Synthesis of chiral α-acetoxy-N-acetylamides from chiral pyrimidylalkanols by the oxidative cleavage of pyrimidine ring

Shigehisa Tanji; Yasutaka Kodaka; Takanori Shibata; Kenso Soai

doi:10.3987/com-98-s1

Synthesis of chiral α-acetoxy-N-acetylamides from chiral pyrimidylalkanols by the oxidative cleavage of pyrimidine ring

Shigehisa Tanji, Yasutaka Kodaka, Takanori Shibata, Kenso Soai^*

^*Corresponding author for this work

Research output: Contribution to journal › Article › peer-review

8 Citations (Scopus)

Abstract

Acetates of chiral 5-pyrimidylalkanols are transformed into chiral α- acetoxy-N-acetylamides and α-acetoxyamides without racemization in high total yields by the oxidative cleavage of pyrimidine ring using ruthenium tetroxide.

Original language	English
Pages (from-to)	151-158
Number of pages	8
Journal	Heterocycles
Volume	52
Issue number	1
DOIs	https://doi.org/10.3987/com-98-s1
Publication status	Published - 2000 Jan 1
Externally published	Yes

ASJC Scopus subject areas

Analytical Chemistry
Pharmacology
Organic Chemistry

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title = "Synthesis of chiral α-acetoxy-N-acetylamides from chiral pyrimidylalkanols by the oxidative cleavage of pyrimidine ring",

abstract = "Acetates of chiral 5-pyrimidylalkanols are transformed into chiral α- acetoxy-N-acetylamides and α-acetoxyamides without racemization in high total yields by the oxidative cleavage of pyrimidine ring using ruthenium tetroxide.",

author = "Shigehisa Tanji and Yasutaka Kodaka and Takanori Shibata and Kenso Soai",

year = "2000",

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doi = "10.3987/com-98-s1",

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publisher = "Japan Institute of Heterocyclic Chemistry",

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AU - Tanji, Shigehisa

AU - Kodaka, Yasutaka

AU - Shibata, Takanori

AU - Soai, Kenso

PY - 2000/1/1

Y1 - 2000/1/1

N2 - Acetates of chiral 5-pyrimidylalkanols are transformed into chiral α- acetoxy-N-acetylamides and α-acetoxyamides without racemization in high total yields by the oxidative cleavage of pyrimidine ring using ruthenium tetroxide.

AB - Acetates of chiral 5-pyrimidylalkanols are transformed into chiral α- acetoxy-N-acetylamides and α-acetoxyamides without racemization in high total yields by the oxidative cleavage of pyrimidine ring using ruthenium tetroxide.

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DO - 10.3987/com-98-s1

M3 - Article

AN - SCOPUS:0033957185

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VL - 52

SP - 151

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JO - Heterocycles

JF - Heterocycles

IS - 1

ER -

Synthesis of chiral α-acetoxy-N-acetylamides from chiral pyrimidylalkanols by the oxidative cleavage of pyrimidine ring

Abstract

ASJC Scopus subject areas

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